1. Signaling Pathways
  2. GPCR/G Protein
    Neuronal Signaling
  3. Opioid Receptor
  4. δ Opioid Receptor/DOR Isoform
  5. δ Opioid Receptor/DOR Activator

δ Opioid Receptor/DOR Activator

δ Opioid Receptor/DOR Activator (1):

Cat. No. Product Name Effect Purity
  • HY-120613
    BMS-986187
    Activator 98.93%
    BMS-986187 is an δ-opioid receptor-selective positive allosteric modulator (PAM) with an EC50 of 0.03 μM and a pKB?of 6.02 (~1?μM). BMS-986187 has no observable PAM activity at the?μ-receptor (EC50=3 μM).